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Substance Name: Xamoterol fumarate [USAN]
RN: 90730-93-1
InChIKey: QEDVGROSOZBGOZ-WXXKFALUSA-N

Note

  • A selective beta-1-adrenergic partial agonist. Because it is a partial agonist (DRUG PARTIAL AGONISM) it acts like an agonist when sympathetic activity is low and as an antagonist when sympathetic activity is high. It reduces MYOCARDIAL ISCHEMIA and improves ventricular function in patients with mild to moderate heart failure. In patients with severe heart failure it has been shown to produce benefits in systolic and diastolic function.

Molecular Weight

  • 794.8506
 

Classification Code

  • Stimulant (Cardiac)
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Names and Synonyms

Name of Substance

  • Xamoterol fumarate [USAN]

Synonyms

  • (+-)-N-(2-((2-Hydroxy-3-(p-hydroxyphenoxy)propyl)amino)ethyl)-4-morpholinecarboxamide fumarate (2:1) (salt)
  • 4-Morphinolinecarboxamide, N-(2-((2-hydroxy-3-(4-hydroxyphenoxy)propyl)amino)ethyl)-, (+-)-, (E)-2-butenedioate (2:1) (salt)
  • ICI 118,587
  • Xamoterol fumarate

Registry Numbers

CAS Registry Number

  • 90730-93-1

System Generated Number

  • 0090730931

Structure Descriptors

InChI

1S/2C16H25N3O5.C4H4O4/c2*20-13-1-3-15(4-2-13)24-12-14(21)11-17-5-6-18-16(22)19-7-9-23-10-8-19;5-3(6)1-2-4(7)8/h2*1-4,14,17,20-21H,5-12H2,(H,18,22);1-2H,(H,5,6)(H,7,8)/b;;2-1+

InChIKey

QEDVGROSOZBGOZ-WXXKFALUSA-N